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Check Intently (1)mitotane decreases amounts of diazepam by affecting hepatic/intestinal enzyme CYP3A4 metabolism. Use Caution/Check. Mitotane is a strong inducer of cytochrome P-4503A4; watch when coadministered with CYP3A4 substrates for probable dosage changes.Administration of benzodiazepines or other drugs that greatly enhance GABAergic inhibi